DOI: 10.1055/s-00000131

Synfacts

Issue 12 · Volume 2010 · December 2010 DOI: 10.1055/s-002-21480

Synform

A94
Zanda, Matteo: SYNFORM ISSUE 2010/11

Synthesis of Natural Products and Potential Drugs

z1327
All PDFs of this category
1327
Rueping, M.; Stoeckel, M.; Sugiono, E.; Theissmann, T.: Synthesis of (R)-Ofloxacin
1328
Beng, T. K.; Gawley, R. E.: Synthesis of (S)-(-)-Ropivacaine
1329
Shimada, N.; Hanari, T.; Kurosaki, Y.; Takeda, K.; Anada, M.; Nambu, H.; Shiro, M.; Hashimoto, S.: Synthesis of endo-6-Aryl-8-oxabicyclo-[3.2.1]oct-3-en-2-one
1330
McGowan, M. A.; Stevenson, C. P.; Schiffler, M. A.; Jacobsen, E. N.: Synthesis of (+)-Peloruside A
1331
Hoye, T. R.; Jeon, J.; Kopel, L. C.; Ryba, T. D.; Tennakoon, M. A.; Wang, Y.: Synthesis of (+)-Peloruside A
1332
al., D. K. Leahy et: Synthesis of BMS-764459
1333
Oelke, A. J.; France, D. J.; Hofmann, T.; Wuitschik, G.; Ley, S. V.: Total Synthesis of Chloptosin
1334
Cheng, B.; Sunderhaus, J. D.; Martin, S. F.: Synthesis of (±)-Pseudotabersonine
1335
Lian, Y.; Miller, L. C.; Born, S.; Sarpong, R.; Davies, H. M. L.: Synthesis of (+)-Barekoxide and (-)-Barekol
1336
Wang, X.-j.; Xu, Y.; Zhang, L.; Krishnamurthy, D.; Wirth, T.; Nicola, T.; Senanayake, C. H.: Synthesis of an LFA-1 Inhibitor
1337
Steinhuebel, D. P.; Krska, S. W.; Alorati, A.; Baxter, J. M.; Belyk, K.; Bishop, B.; Palucki, M.; Sun, Y.; Davies, I. W.: Synthesis of Telcagepant
1338
Sohn, T.-i.; Kim, M. J.; Kim, D.: Synthesis of Trilobacin
1339
Simmons, E. M.; Hardin-Narayan, A. R.; Guo, X.; Sarpong, R.: Formal Synthesis of (±)-Cortistatin A
1340
Ripin, D. H. Brown; al., D. S. Teager et: Synthesis of Tenofovir Disoproxil Fumarate

Synthesis of Heterocycles

z1341
All PDFs of this category
1341
Desai, A. A.; Wulff, W. D.: Synthesis of Chiral Aziridines from Imines and Diazoacetamides
1342
Shimizu, R.; Egami, H.; Nagi, T.; Chae, J.; Hamashima, Y.; Sodeoka, M.: Direct C2 Indole Trifluoromethylation Using Togni’s Reagent
1343
Baeza, A.; Mendiola, J.; Burgos, C.; Alvares-Builla, J.; Vaquero, J. J.: Synthesis of Pyridopyrrolopyrimidines. Total Synthesis of Varioline B and Deoxyvariolin B
1344
Akkilagunta, V. K.; Reddy, V. P.; Kakulapati, R. R.: Synthesis of Quinoxalines via Ru/C Benzoin Oxidation and Diamine Condensation
1345
Zhang, X.; Teo, W. T.; Sally; Chan, P. W. H.: Facile Acid-Catalyzed Route to Thiazoles from Propargylic Alcohols and Thioamides
1346
Hong, D.; Chen, Z.; Lin, X.; Wang, Y.: Synthesis of Indoles from 2-Azidoacrylate and ortho-Silyl Aryltriflates
1347
Ballini, R.; Gabrielli, S.; Palmieri, A.: Synthesis of Tetrasubstituted Furans by Michael Addition to β-Nitroacrylates
1348
Toyoshima, T.; Mikano, Y.; Miura, T.; Murakami, M.: Palladium-Catalyzed Synthesis of 3,3-Disubstituted Oxindoles
1349
Barluenga, J.; Lonzi, G.; Riesgo, L.; López, L. A.; Tomás, M.: Copper(I)-Catalyzed Annulation Route to Indolizines
1350
Wray, B. C.; Stambuli, J. P.: Synthesis of N-Arylindazoles and Benz-imidazoles from ortho-Aminobenzoximes
1351
Inman, M.; Moody, C. J.: Copper-Mediated Synthesis of Indolequinones from Bromoquinones
1352
Yang, Q.; Cao, H.; Robertson, A.; Alper, H.: Palladium-Catalyzed Cyclocarbonylative Synthesis of Dibenzoxazepinones
1353
Fujita, M.; Yoshida, Y.; Miyata, K.; Wakisaka, A.; Sugimura, T.: Enantioselective Synthesis of Dihydro-isochromanones Using Hypervalent Iodine
1354
Kwok, S. W.; Fotsing, J. R.; Fraser, R. J.; Rodionov, V. O.; Fokin, V. V.: Synthesis of 1,5-Diaryl-1,2,3-triazoles Under Transition-Metal-Free Conditions
1355
Zeghida, W.; Besnard, C.; Lacour, J.: Rhodium(II)-Catalyzed Synthesis of Polyether Macrocyles

Synthesis of Materials and Unnatural Products

z1357
All PDFs of this category
1357
Sun, Z.; Huang, K.-W.; Wu, J.: Soluble and Stable Zethrenebis(carboximide) and Its Quinone
1358
Mori, H.; Tando, I.; Tanaka, H.: Alternating Copolymers of Anthracene via Novel Radical ROP
1359
Jakob, S.; Moreno, A.; Zhang, X.; Bertschi, L.; Smith, P.; Schlüter, A. D.; Sakamoto, J.: Unsubstituted Polyphenylenes via a ‘Shaving’ Approach
1360
Zhang, H.-j.; Wei, J.; Zhao, F.; Liang, Y.; Wang, Z.; Xi, Z.: Highly Selective Synthesis of Dibenzo[a,c]cyclooctatetraenes
1361
Criado, A.; Gómez-Escalonilla, M. J.; Fierro, J. L. G.; Urbina, A.; Peña, D.; Guitián, E.; Langa, F.: A New Functionalization Method of SWCNTs through Cycloaddition
1362
Chen, J.-D.; Lu, H.-Y.; Chen, C.-F.: Scale Up, Spice Up
1363
Nakanishi, W.; Hitosugi, S.; Piskareva, A.; Shimada, Y.; Taka, H.; Kita, H.; Isobe, H.: Efficient Bipolar Transport Material for OLEDs
1364
Xiao, Z.; Matsuo, Y.; Nakamura, E.: Annulated Fullerenes
1365
Appel, E. A.; Biedermann, F.; Rauwald, U.; Jones, S. T.; Zayed, J. M.; Scherman, O. A.: Hosting Hydrogel Formation
1366
Sessler, J. L.; Cai, J.; Gong, H.-Y.; Yang, X.; Arambula, J. F.; Hay, B. P.: One Scaffold, Different Motifs
1367
Harvey, P. D.; al., W.-Y. Wong et: Light-Emitting Platinum-Containing Polymers
1368
Petrov, A. R.; Daniliuc, C. G.; Jones, P. G.; Tamm, M.: A New Route to Diaminoacetylenes
1369
Proń, A.; Baumgarten, M.; Müllen, K.: Phenylene-Bridged Boron-Nitrogen Containing Dendrimers
1370
Fischer, F. R.; Nuckolls, C.: Alkyne ROMP: ‘It’s Alive!!!’

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z1371
All PDFs of this category
1371
Ikeda, M.; Miyake, Y.; Nishibayashi, Y.: Cooperative Ruthenium and Organocatalysis
1372
Hou, G.; Li, W.; Ma, M.; Zhang, X.: Iridium-Catalyzed Asymmetric Hydrogenation of Unprotected β-Enamine Esters
1373
Nishimura, T.; Maeda, Y.; Hayashi, T.: Asymmetric Cyclopropanation Using Dimethyl Diazomalonate
1374
Tsoi, Y.-T.; Zhou, Z.; Chan, A. S. C.; Yu, W.-Y.: Stereoselective Synthesis of (E)-α,β-Diarylacrylates
1375
Zheng, K.; Yang, Y.; Zhao, J.; Yin, C.; Lin, L.; Liu, X.; Feng, X.: Solvent-Free Magnesium-Catalyzed Enantioselective Ketone-Ene Reactions
1376
Chen, X.; Zhu, Y.; Qiao, Z.; Xie, M.; Lin, L.; Liu, X.; Feng, X.: Nickel-Catalyzed Aldol Reaction Between α-Isothiocyanato Imide and Aldehydes
1377
Wang, Z.; Chen, D.; Yang, Z.; Bai, S.; Liu, X.; Lin, L.; Feng, X.: Catalytic Asymmetric Michael Addition to 4-Oxo-4-arylbutenoates
1378
Landert, H.; Spindler, F.; Wyss, A.; Blaser, H.-U.; Pugin, B.; Ribourduoille, Y.; Gschwend, B.; Ramalingam, B.; Pfaltz, A.: New Chiral Bidentate Secondary Phosphine Oxide Ligands for Hydrogenation
1379
Antonchick, A. P.; Gerding-Reimers, C.; Catarinella, M.; Schürmann, M.; Preut, H.; Ziegler, S.; Rauh, D.; Waldmann, H.: Enantioselective Synthesis of Spirooxindoles Inspired by Natural Products
1380
Morgen, M.; Bretzke, S.; Li, P.; Menche, D.: Synthesis of 1,3-syn and -anti-Tetrahydro-pyrimidinones
1381
Ito, J.-i.; Asai, R.; Nishiyama, H.: Asymmetric Ru-Phebox Catalyzed Alkynylation
1382
Zhu, S.; Xu, X.; Perman, J.; Zhang, X. P.: Cobalt(II)-Catalyzed Stereoselective Cyclopropanation of Alkenes
1383
Yeh, M.-C. P.; Lin, M.-N.; Chang, W.-J.; Liou, J.-L.; Shih, Y.-F.: Gold(I)-Catalyzed Diastereoselective Pyrrolidine Synthesis
1384
Nishimura, T.; Makino, H.; Nagaosa, M.; Hayashi, T.: Rhodium-Catalyzed Asymmetric 1,6-Addition of Enynamides
1385
Guo, H.; Herdtweck, E.; Bach, T.: A Lewis Acid Catalyzed Asymmetric Photocycloaddition
1386
Kim, S. J.; Jang, D. O.: Indium-Mediated Enantioselective Allylation
1387
Shintani, R.; Takeda, M.; Tsuji, T.; Hayashi, T.: Asymmetric Arylation of N-Tosyl Ketimines
1388
Sauer, S. J.; Garnsey, M. R.; Coltart, D. M.: Reductive Enolization in Aldol Addition to Enolizable Aldehydes
1389
Fañanás-Mastral, M.; Feringa, B. L.: Copper-Catalyzed Addition of Grignards to Allylic α-Haloacetates
1390
McDonald, R. I.; Wong, G. W.; Neupane, R. P.; Stahl, S. S.; Landis, C. R.: Rhodium-Catalyzed Asymmetric Hydro-formylation
1391
Shao, C.; Yu, H.-J.; Wu, N.-Y.; Feng, C.-G.; Lin, G.-Q.: C1-Symmetric Dicyclopentadienes in Rh-Catalyzed Arylation of N-Tosylarylimines
1392
Teichert, J. F.; Zhang, S.; van Zijl, A. W.; Slaa, J. W.; Minnaard, A. J.; Feringa, B. L.: Chiral N-Heterocycles via Asymmetric Allylic Methylation-Ring-Closing Metathesis
1393
Llaveria, J.; Beltrán, Á.; Díaz-Requejo, M. M.; Matheu, M. I.; Castillón, S.; Pérez, P. J.: Regio- and Stereospecific Aziridinzation of Unsymmetric Conjugated Dienes
1394
Dugal-Tessier, J.; Dake, G. R.; Gates, D. P.: Asymmetric Allylic Alkylation with Phosphaalkene-Oxazoline Ligands
1395
Huang, S.; Petersen, T. B.; Lipshutz, B. H.: Atropselective Biaryl Coupling in the Synthesis of (+)-Korupensamine B
1396
Takebayashi, S.; John, J. M.; Bergens, S. H.: Ruthenium-Catalyzed Asymmetric Monohydrogenation of meso-Cyclic Imides
1397
Moquist, P. N.; Kodama, T.; Schaus, S. E.: Combined Acid System for Asymmetric Addition of Boronates to Chromene Acetals
1398
Hawner, C.; Müller, D.; Gremaud, L.; Felouat, A.; Woodward, S.; Alexakis, A.: Conjugate Addition of Aryl Alanes to Form Quaternary Stereocenters
1399
Zhu, L.; Meng, Q.; Fan, W.; Xie, X.; Zhang, Z.: Ruthenium-Catalyzed Asymmetric Reduction of α-Keto Acids
1400
Zheng, S.; Gao, N.; Liu, W.; Liu, D.; Zhao, X.; Cohen, T.: Synthesis of Enantiopure Allyl Phenyl Sulfides

Metal-Mediated Synthesis

z1401
All PDFs of this category
1401
Maji, M. S.; Murarka, S.; Studer, A.: Metal-Free Coupling of Aryl and Alkynyl Grignard Reagents Mediated by TEMPO
1402
Ishizuka, K.; Seike, H.; Hatakeyama, T.; Nakamura, M.: Alkenylative Cross-Coupling between Alkyl Sulfides and Grignard Reagents
1403
Ohmura, T.; Awano, T.; Suginome, M.: Stereospecific Suzuki Coupling with Inversion of Stereoconfiguration
1404
Lu, Z.; Fu, G. C.: Csp³-Csp³ Suzuki Cross-Coupling Using Unactivated Secondary Alkyl Chlorides
1405
Molander, G. A.; Beaumard, F.: Nickel-Catalyzed C-O Activation of Phenol Derivatives
1406
Kyne, R. E.; Ryan, M. C.; Kliman, L. T.; Morken, J. P.: Allylation of Nitrosobenzene with Pinacol Allylboronates
1407
Duan, H.; Meng, L.; Bao, D.; Zhang, H.; Li, Y.; Lei, A.: ZnCl2-Enhanced Negishi Coupling of Secondary Benzyl Trifluoroacetates
1408
Fandrick, K. R.; Fandrick, D. R.; Gao, J. J.; Reeves, J. T.; Tan, Z.; Li, W.; Song, J. J.; Lu, B.; Yee, N. K.; Senanayake, C. H.: Zinc Alkoxide Catalyzed Allylations of Ketones with Allyl Pinacol Boronates
1409
Renaudat, A.; Jean-Gérard, L.; Jazzar, R.; Kefalidis, C. E.; Clot, E.; Baudoin, O.: Palladium-Catalyzed β-Arylation of Carboxylic Esters
1410
Gao, K.; Lee, P.-S.; Fujita, T.; Yoshikai, N.: Cobalt-Catalyzed Hydroarylation of Alkynes Through C-H Bond Activation
1411
Dickschat, A.; Studer, A.: Radical Addition of Arylboronic Acids to Olefins
1412
Shirokane, K.; Kurosaki, Y.; Sato, T.; Chida, N.: Nucleophilic Addition to N-Methoxyamides via N-Oxyiminium Ions
1413
Seiple, I. B.; Su, S.; Rodriguez, R. A.; Gianatassio, R.; Fujiwara, Y.; Sobel, A. L.; Baran, P. S.: C-H Arylation of N-Heterocycles with Arylboronic Acids
1414
Pintaric, C.; Olivero, S.; Gimbert, Y.; Chavant, P. Y.; Duñach, E.: Catalytic Magnesium in Direct Coupling of Benzylic Halides with Pinacolborane
1415
Reeves, J. T.; Fandrick, D. R.; Tan, Z.; Song, J. J.; Lee, H.; Yee, N. K.; Senanayake, C. H.: Cross-Coupling of Aryltrimethylammonium Triflates with Aryl Grignard Reagents

Organo- and Biocatalysis

z1417
All PDFs of this category
1417
Holloway, C. A.; Muratore, M. E.; Storer, R. I.; Dixon, D. J.: Brønsted Acid Catalyzed Pictet-Spengler Cyclization of Keto Acids
1418
Kavanagh, S. A.; Piccinini, A.; Connon, S. J.: Organocatalytic Corey-Chaykovsky Reaction of Ketones
1419
Neumann, M.; Füldner, S.; König, B.; Zeitler, K.: Organophotoredox Catalysis
1420
Urushima, T.; Sakamoto, D.; Ishikawa, H.; Hayashi, Y.: One-Pot Synthesis of Chiral Piperidines Using Diphenylprolinol Silyl Ether
1421
Wang, X.-F.; Hua, Q.-L.; Cheng, Y.; An, X.-L.; Yang, Q.-Q.; Chen, J.-R.; Xiao, W.-J.: Sulfa-Michael Reaction Cascade for the Synthesis of Chromans
1422
Liu, Y.-L.; Wang, B.-L.; Cao, J.-J.; Chen, L.; Zhang, Y.-X.; Wang, C.; Zhou, J.: Asymmetric Morita-Baylis-Hillman Reactions of Acrolein
1423
Park, S. E.; Nam, E. H.; Jang, H. B.; Oh, J. S.; Some, S.; Lee, Y. S.; Song, C. E.: Highly Efficient Desymmetrization of Glutaric Anhydrides
1424
Shao, P.-L.; Chen, X.-Y.; Ye, S.: Formal [3+2] Cycloaddition of Ketenes and Oxaziridines
1425
Jiang, H.; Gschwend, B.; Albrecht, Ł.; Jørgensen, K. A.: Practical Enantioselective One-Pot Syntheses of β-Hydroxy and β-Amino Esters
1426
Klauber, E. G.; De, C. Kanta; Shah, T. K.; Seidel, D.: Asymmetric Anion Binding DMAP Catalysis in the Kinetic Resolution of Propargylic Amines
1427
Dohi, T.; Takenaga, N.; Fukushima, K.-i.; Uchiyama, T.; Kato, D.; Motoo, S.; Fujioka, H.; Kita, Y.: Hypervalent Iodine(III) Organocatalysts
1428
Cai, Q.; Zheng, C.; You, S.-L.: Intramolecular Aza-Michael Addition of Indoles
1429
Jin, J.; Oskam, P. C.; Karmee, S. K.; Straathof, A. J. J.; Hanefeld, U.: A Bifunctional Enzyme for a Michael Addition-Oxidation Sequence

Polymer-Supported Synthesis

z1431
All PDFs of this category
1431
Park, C. P.; Kim, D.-P.: A Flow Reaction System Using Catalytic Magnetic Particles
1432
Audic, N.; Dyer, P. W.; Hope, E. G.; Stuart, A. M.; Suhard, S.: Perfluoroalkylated Polymer-Supported Palladium Catalyst
1433
Chen, Z.; Cui, Z.-M.; Niu, F.; Jiang, L.; Song, W.-G.: Palladium Nanoparticles in Silica Hollow Spheres with Mesoporous Walls
1434
Zeng, T.; Song, G.; Moores, A.; Li, C.-J.: Cross-Dehydrogenative Coupling with Fe3O4 Nanoparticles
1435
Xu, W.-M.; He, J.; Yu, M.-Q.; Shen, G.-X.: Modification of a Vitamin D Analogue Using a Supported Selenium Reagent
1436
Rajagopal, G.; Selvaraj, S.; Dhahagani, K.: Asymmetric Cyanosilylation with Supported Cu(II) Salen Complexes
1437
Yamazaki, K.; Kawamorita, S.; Ohmiya, H.; Sawamura, M.: ortho-Borylation of Phenols with Silica-SMAP-Ir
1438
Ricci, A.; Bernardi, L.; Gioia, C.; Vierucci, S.; Robitzer, M.; Quignard, F.: Asymmetric Aldol Reaction in Water Catalyzed by Chitosan Aerogel
1439
Yamada, Y. M. A.; Watanabe, T.; Beppu, T.; Fukuyama, N.; Torii, K.; Uozumi, Y.: Suzuki-Miyaura Couplings with Palladium Membrane Installed Microreactors
1440
Dhakshinamoorthy, A.; Alvaro, M.; Garcia, H.: An Iron Metal-Organic Framework Catalyst for Thiol Oxidation
1441
Mikami, Y.; Noujima, A.; Mitsudome, T.; Mizugaki, T.; Jitsukawa, K.; Kaneda, K.: Deoxygenation of Epoxides with Hydrotalcite-Supported Silver Nanoparticles
1442
Takeda, K.; Oohara, T.; Anada, M.; Nambu, H.; Hashimoto, S.: Asymmetric C-H Insertion with a Polymer-Supported Rhodium Complex
1443
Okudomi, M.; Ageishi, K.; Yamada, T.; Chihara, N.; Nakagawa, T.; Mizuochi, K.; Matsumoto, K.: Enantioselective Hydrolysis of Soluble Polymer-Supported Carboxylates