DOI: 10.1055/s-00000083

Synlett

Ausgabe 20 · Volume 28 · Dezember 2017 DOI: 10.1055/s-007-35789

editorial

  • I

    Editorial

    • account

  • 2685
    Quiclet-Sire, Béatrice; Zard, Samir Z.:

    Convergent Routes to Pyrroles Exploiting the Unusual Radical Chemistry of Xanthates – An Overview

    Image for article: Convergent Routes to Pyrroles Exploiting the Unusual Radical Chemistry of Xanthates – An Overview
  • 2697
    Davies, Stephen G.; Fletcher, Ai M.; Roberts, Paul M.; Thomson, James E.:

    Asymmetric Synthesis of Pyrrolizidines, Indolizidines and Quinolizidines via a Double Reductive Cyclisation Protocol

    Image for article: Asymmetric Synthesis of Pyrrolizidines, Indolizidines and Quinolizidines via a Double Reductive Cyclisation Protocol
  • 2707
    Shaaban, Saad; Maulide, Nuno:

    Metal-Free Redox Transformations for C–C and C–N Bond Construction

    Image for article: Metal-Free Redox Transformations for C–C and C–N Bond Construction
  • 2714
    Liu, Wenbo; Li, Chao-Jun:

    Recent Synthetic Applications of Catalyst-Free Photochemistry

    Image for article: Recent Synthetic Applications of Catalyst-Free Photochemistry

    • letter

  • 2755
    Thullen, Scott M.; Rubush, David M.; Rovis, Tomislav:

    A Photochemical Two-Step Formal [5+2] Cycloaddition: A Condensation–Ring-Expansion Approach to Substituted Azepanes

    Image for article: A Photochemical Two-Step Formal [5+2] Cycloaddition: A Condensation–Ring-Expansion Approach to Substituted Azepanes
    Supporting Information (PDF)
  • 2759
    Vásquez-Céspedes, Suhelen; Holtkamp, Michael; Karst, Uwe; Glorius, Frank:

    Reusable and Magnetic Palladium and Copper Oxide Catalysts in Direct ortho and meta Arylation of Anilide Derivatives

    Image for article: Reusable and Magnetic Palladium and Copper Oxide Catalysts in Direct <i>ortho</i> and <i>meta</i> Arylation of Anilide Derivatives
    Supporting Information (PDF)
  • 2765
    Aeyad, Tahani; Williams, Jason D.; Meijer, Anthony J. H. M.; Coldham, Iain:

    Lithiation–Substitution of N-Boc-2-phenylazepane

    Image for article: Lithiation–Substitution of <i>N</i>-Boc-2-phenylazepane
    Supporting Information (PDF)
  • 2769
    Piras, Monica; Andriu, Alexandra; Testa, Andrea; Wienecke, Paul; Fleming, Ian N.; Zanda, Matteo:

    Design and Synthesis of an RGD Peptidomimetic-Paclitaxel Conjugate Targeting αvβ3 Integrin for Tumour-Directed Drug Delivery

    Image for article: Design and Synthesis of an RGD Peptidomimetic-Paclitaxel Conjugate Targeting α<sub>v</sub>β<sub>3</sub> Integrin for Tumour-Directed Drug Delivery
    Supporting Information (PDF)
  • 2777
    Chen, Jun; Lu, Lingxiao; Wulff, Jeremy E.:

    Radical Stabilization Algorithm as a Predictive Tool for Novel and Reported Noncanonical Thiele’s Acid Analogues

    Image for article: Radical Stabilization Algorithm as a Predictive Tool for Novel and Reported Noncanonical Thiele’s Acid Analogues
    Supporting Information (PDF)
  • 2783
    Schleper, A. Lennart; Voll, Constantin-Christian A.; Engelhart, Jens U.; Swager, Timothy M.:

    Iptycene-Containing Azaacenes with Tunable Luminescence

    Image for article: Iptycene-Containing Azaacenes with Tunable Luminescence
    Supporting Information (PDF)
  • 2790
    Bagdžiūnas, Gintautas; Stončius, Sigitas; Butkus, Eugenijus:

    Synthesis of Star-Shaped Aromatic Derivatives with Chirality Predetermined by Bicyclo[3.3.1]nonane Framework

    Image for article: Synthesis of Star-Shaped Aromatic Derivatives with Chirality Predetermined by Bicyclo[3.3.1]nonane Framework
    Supporting Information (PDF)
  • 2795
    Afsar, Ashfaq; Cowell, Joseph; Distler, Petr; Harwood, Laurence M.; John, Jan; Westwood, James:

    Synthesis of Novel BTPhen-Functionalized Silica-Coated Magnetic Nanoparticles for Separating Trivalent Actinides and Lanthanides

    Image for article: Synthesis of Novel BTPhen-Functionalized Silica-Coated Magnetic Nanoparticles for Separating Trivalent Actinides and Lanthanides
    Supporting Information (PDF)
  • 2800
    Chernichenko, Nataliya M.; Shevchuk, Vadim N.; Averin, Alexei D.; Maloshitskaya, Olga A.; Beletskaya, Irina P.:

    Synthesis of Dansyl-Substituted Cryptands Containing Triaza­cycloalkane Moieties and their Evaluation as Fluorescent Chemosensors

    Image for article: Synthesis of Dansyl-Substituted Cryptands Containing Triaza­cycloalkane Moieties and their Evaluation as Fluorescent Chemosensors
    Supporting Information (PDF)
  • 2807
    Chui, Tin-Ki; Chow, Hak-Fun:

    New Triazole-Containing Branched Bis(dipeptidomimetic) – Switching from Self-Dimerization to Anion-Binding Properties

    Image for article: New Triazole-Containing Branched Bis(dipeptidomimetic) – Switching from Self-Dimerization to Anion-Binding Properties
    Supporting Information (PDF)
  • 2812
    Ichioka, Fumiki; Itai, Yuhei; Nishii, Yuji; Miura, Masahiro:

    Palladium-Catalyzed Direct C2-Arylation of Benzo[b]thiophenes with Electron-Rich Aryl Halides: Facile Access to Thienoacene Derivatives

    Image for article: Palladium-Catalyzed Direct C2-Arylation of Benzo[<i>b</i>]thiophenes with Electron-Rich Aryl Halides: Facile Access to Thienoacene Derivatives
    Supporting Information (PDF)
  • 2817
    Ketels, Marthe; Ziegler, Dorothée S.; Knochel, Paul:

    Selective Zincation of 1,2-Dicyanobenzene and Related Benzonitriles in Continuous Flow Using In Situ Trapping Metalations

    Image for article: Selective Zincation of 1,2-Dicyanobenzene and Related Benzonitriles in Continuous Flow Using In Situ Trapping Metalations
    Supporting Information (PDF)
  • 2823
    Hamel, Jean-Denys; Beaudoin, Meggan; Cloutier, Mélissa; Paquin, Jean-François:

    Hydrogen-Bond-Promoted Friedel–Crafts Reaction of Secondary Propargylic Fluorides: Preparation of 1-Alkyl-1-aryl-2-alkynes

    Image for article: Hydrogen-Bond-Promoted Friedel–Crafts Reaction of Secondary Propargylic Fluorides: Preparation of 1-Alkyl-1-aryl-2-alkynes
    Supporting Information (PDF)
  • 2829
    Gao, Ang; Liu, Xiu-Yan; Ding, Chang-Hua; Hou, Xue-Long:

    Diastereoselective Palladium-Catalyzed Conjugate Addition of Arylboronic Acids to α-Substituted Cyclic Enones

    Image for article: Diastereoselective Palladium-Catalyzed Conjugate Addition of Arylboronic Acids to α-Substituted Cyclic Enones
    Supporting Information (PDF)
  • 2833
    Benoit, Emeline; Dansereau, Julien; Gagnon, Alexandre:

    Palladium-Catalyzed Carbonylative Cross-Coupling Reaction between Aryl(Heteroaryl) Iodides and Tricyclopropylbismuth: Expedient Access to Aryl Cyclopropylketones

    Image for article: Palladium-Catalyzed Carbonylative Cross-Coupling Reaction between Aryl(Heteroaryl) Iodides and Tricyclopropylbismuth: Expedient Access to Aryl Cyclopropylketones
    Supporting Information (PDF)
  • 2839
    Xu, Lanting; Tan, Lushi; Ma, Dawei:

    Rhodium-Catalyzed Regioselective C7-Functionalization of Indole Derivatives with Acrylates by Using an N-Imino Directing Group

    Image for article: Rhodium-Catalyzed Regioselective C7-Functionalization of Indole Derivatives with Acrylates by Using an N-Imino Directing Group
    Supporting Information (PDF)
  • 2845
    Corbett, Michael T.; Caille, Seb:

    A Bench-Stable Vilsmeier Reagent for in situ Alcohol Activation: Synthetic Application in the Synthesis of 2-Amino-2-Thiazolines

    Image for article: A Bench-Stable Vilsmeier Reagent for in situ Alcohol Activation: Synthetic Application in the Synthesis of 2-Amino-2-Thiazolines
    Supporting Information (PDF)
  • 2851
    Isbrandt, Eric S.; Vandavasi, Jaya Kishore; Zhang, Wanying; Jamshidi, Mohammad P.; Newman, Stephen G.:

    Catalytic Deuteration of Aldehydes with D2O

    Image for article: Catalytic Deuteration of Aldehydes with D<sub>2</sub>O
    Supporting Information (PDF)
  • 2855
    Labes, Ricardo; González-Calderón, Davir; Battilocchio, Claudio; Mateos, Carlos; Cumming, Graham R.; de Frutos, Oscar; Rincón, Juan A.; Ley, Steven V.:

    Rapid Continuous Ruthenium-Catalysed Transfer Hydrogenation of Aromatic Nitriles to Primary Amines

    Image for article: Rapid Continuous Ruthenium-Catalysed Transfer Hydrogenation of Aromatic Nitriles to Primary Amines
    Open Access
    Supporting Information (PDF)
  • 2859
    Irwin, Lauren C.; Kerr, Michael A.:

    One-Pot Michael Addition/Radical Cyclization Reaction of N-Acryloyl Indoles

    Image for article: One-Pot Michael Addition/Radical Cyclization Reaction of <i>N</i>-Acryloyl Indoles
    Supporting Information (PDF)
  • 2865
    Ramadhar, Timothy R.; Kawakami, Jun-ichi; Batey, Robert A.:

    Sequential O-Arylation/Lanthanide(III)-Catalyzed [3,3]-Sigmatropic Rearrangement of Bromo-Substituted Allylic Alcohols

    Image for article: Sequential O-Arylation/Lanthanide(III)-Catalyzed [3,3]-Sigmatropic Rearrangement of Bromo-Substituted Allylic Alcohols
    Supporting Information (PDF)
  • 2871
    Eljo, Jasmin; Carle, Myriam S.; Murphy, Graham K.:

    Hypervalent Iodine-Based Activation of Triphenylphosphine for the Functionalization of Alcohols

    Image for article: Hypervalent Iodine-Based Activation of Triphenylphosphine for the Functionalization of Alcohols
    Supporting Information (PDF)
  • 2876
    Zhi, Ying; Zhao, Kun; von Essen, Carolina; Rissanen, Kari; Enders, Dieter:

    Thiourea-Catalyzed Domino Michael–Mannich [3+2] Cycloadditions: A Strategy for the Asymmetric Synthesis of 3,3′-Pyrrolidinyl-dispirooxindoles

    Image for article: Thiourea-Catalyzed Domino Michael–Mannich [3+2] Cycloadditions: A Strategy for the Asymmetric Synthesis of 3,3′-Pyrrolidinyl-dispirooxindoles
    Supporting Information (PDF)
  • 2881
    Papatzimas, James W.; Gorobets, Evgueni; Brownsey, Duncan K.; Maity, Ranjan; Bahlis, Nizar J.; Derksen, Darren J.:

    A General Strategy for the Preparation of Thalidomide-Conjugate Linkers

    Image for article: A General Strategy for the Preparation of Thalidomide-Conjugate Linkers
    Supporting Information (PDF)
  • 2886
    Fahandej-Sadi, Anis; Lundgren, Rylan J.:

    Copper-Mediated Synthesis of Monofluoro Aryl Acetates via Decarboxylative Cross-Coupling

    Image for article: Copper-Mediated Synthesis of Monofluoro Aryl Acetates via Decarboxylative Cross-Coupling
    Supporting Information (PDF)
  • 2891
    Barraza, Scott J.; Denmark, Scott E.:

    Unexpected Rearrangement of 2-Bromoaniline under Biphasic Alkylation Conditions

    Image for article: Unexpected Rearrangement of 2-Bromoaniline under Biphasic Alkylation Conditions
    Supporting Information (PDF)
  • 2896
    Lapinskaite, Ringaile; Ghavre, Mukund; Rintelmann, Chelsea L.; Bedard, Korey; Dela Paz, Helen E.; Hudlicky, Tomas:

    Chemoenzymatic Formal Total Synthesis of Pancratistatin from Narciclasine-Type Compounds via Myers Transposition: Model Study for a Short Conversion of Narciclasine to Pancratistatin

    Image for article: Chemoenzymatic Formal Total Synthesis of Pancratistatin from Narciclasine-Type Compounds via Myers Transposition: Model Study for a Short Conversion of Narciclasine to Pancratistatin
    Supporting Information (PDF)
  • 2901
    Emberson, Kassandra; Tran, Ngan; Metallinos, Costa:

    Diastereoselective Lithiation of N-Benzyl Pyrroloimidazolones Derived from l-Proline Hydantoin

    Image for article: Diastereoselective Lithiation of <i>N</i>-Benzyl Pyrroloimidazolones Derived from <sc>l</sc>-Proline Hydantoin
    Supporting Information (PDF)
  • 2906
    Ma, Zhi-Xiong; Fang, Li-Chao; Haugen, Bryan J.; Bruckbauer, Daniel; Feltenberger, John B.; Hsung, Richard P.:

    Facile Synthesis of 3-Amido-Dienynes via a Tandem α-Propargylation–Isomerization of Chiral Allenamides and their Applications in Diels–Alder Cycloadditions

    Image for article: Facile Synthesis of 3-Amido-Dienynes via a Tandem α-Propargylation–Isomerization of Chiral Allenamides and their Applications in Diels–Alder Cycloadditions
    Supporting Information (PDF)
  • 2913
    Yamamoto, Yasutomo; Yamaguchi, Tatsuya; Kaneshige, Atsunori; Hashimoto, Aiko; Kaibe, Sachiho; Miyawaki, Akari; Yamada, Ken-ichi; Tomioka, Kiyoshi:

    Consecutive Aminolithiation–Carbolithiation of a Linear Aminoalkene Bearing Terminal Vinyl Sulfide Moiety to Give Hydro­indolizine

    Image for article: Consecutive Aminolithiation–Carbolithiation of a Linear Aminoalkene Bearing Terminal Vinyl Sulfide Moiety to Give Hydro­indolizine
    Supporting Information (PDF)
  • 2918
    Jia, Zhi-Jun; Merten, Christian; Knauer, Lena; Murarka, Sandip; Strohmann, Carsten; Waldmann, Herbert:

    Biology-Oriented Synthesis of Decahydro-4,8-epoxyazulene Scaffolds

    Image for article: Biology-Oriented Synthesis of Decahydro-4,8-epoxyazulene Scaffolds
    Supporting Information (PDF)
  • 2923
    Onge, Brent St.; Green, James R.:

    Nicholas Reactions of Alkynyl- and Alkenyltrifluoroborates

    Image for article: Nicholas Reactions of Alkynyl- and Alkenyltrifluoroborates
    Supporting Information (PDF)
  • 2928
    Cooze, Christopher; Manchoju, Amarender; Pansare, Sunil V.:

    Synthesis of (–)-Muricatacin and (–)-(R,R)-L-Factor Involving an Organocatalytic Direct Vinylogous Aldol Reaction

    Image for article: Synthesis of (–)-Muricatacin and (–)-(<i>R</i>,<i>R</i>)-L-Factor Involving an Organocatalytic Direct Vinylogous Aldol Reaction
    Supporting Information (PDF)
  • 2933
    Wang, Tao; Oswood, Christian J.; Hoye, Thomas R.:

    Trapping of Hexadehydro-Diels–Alder Benzynes with Exocyclic, Conjugated Enals as a Route to Fused Spirocyclic Benzopyran Motifs

    Image for article: Trapping of Hexadehydro-Diels–Alder Benzynes with Exocyclic, Conjugated Enals as a Route to Fused Spirocyclic Benzopyran Motifs
    Supporting Information (PDF)
  • 2936
    Nambo, Masakazu; Yim, Jacky C.-H.; Fowler, Kevin G.; Crudden, Cathleen M.:

    Synthesis of Tetraarylmethanes by the Triflic Acid-Promoted Formal Cross-Dehydrogenative Coupling of Triarylmethanes with Arenes

    Image for article: Synthesis of Tetraarylmethanes by the Triflic Acid-Promoted Formal Cross-Dehydrogenative Coupling of Triarylmethanes with Arenes
    Supporting Information (PDF)
  • 2941
    Morimoto, Koji; Koseki, Doichi; Dohi, Toshifumi; Kita, Yasuyuki:

    Oxidative Biaryl Coupling of N-Aryl Anilines by Using a Hypervalent Iodine(III) Reagent

    Image for article: Oxidative Biaryl Coupling of <i>N</i>-Aryl Anilines by Using a Hypervalent Iodine(III) Reagent
  • 2946
    Mohr, Lisa-Marie; Bach, Thorsten:

    Intermolecular [2+2] Photocycloaddition of β-Nitrostyrenes to Olefins upon Irradiation with Visible Light

    Image for article: Intermolecular [2+2] Photocycloaddition of β-Nitrostyrenes to Olefins upon Irradiation with Visible Light
    Open Access
    Supporting Information (PDF) Primary Data (ZIP)
  • 2951
    Hurtak, Jessica A.; McDonald, Frank E.:

    Regioselectivity of Mercury-Promoted Oxacyclizations of Alkynyl Diols

    Image for article: Regioselectivity of Mercury-Promoted Oxacyclizations of Alkynyl Diols
    Supporting Information (PDF)
  • 2956
    Gao, Ke; Yamamoto, Keita; Nogi, Keisuke; Yorimitsu, Hideki:

    Palladium-Catalyzed Arylation of Benzylic C–H Bonds of Azaarylmethanes with Aryl Sulfides

    Image for article: Palladium-Catalyzed Arylation of Benzylic C–H Bonds of Azaarylmethanes with Aryl Sulfides
    Supporting Information (PDF)
  • 2961
    Narayanappa, Arkesh; Hurem, David; McNulty, James:

    Regioselective Ylide Formation on Acetal-Functionalized Trialkyl Phosphonium Salts: Extending the Scope of Carbonyl Homologation

    Image for article: Regioselective Ylide Formation on Acetal-Functionalized Trialkyl Phosphonium Salts: Extending the Scope of Carbonyl Homologation
    Supporting Information (PDF)
  • 2966
    Hirai, Yoshinori; Uozumi, Yasuhiro:

    Preparation of Aryl(dicyclohexyl)phosphines by C–P Bond-Forming Cross-Coupling in Water Catalyzed by an Amphiphilic-Resin-Supported Palladium Complex

    Image for article: Preparation of Aryl(dicyclohexyl)phosphines by C–P Bond-Forming Cross-Coupling in Water Catalyzed by an Amphiphilic-Resin-Supported Palladium Complex
    Supporting Information (PDF)
  • 2971
    Zhao, Changjia; Sibi, Mukund P.:

    Enantioselective and Diastereoselective Conjugate Radical Additions to α-Arylidene Ketones and Lactones

    Image for article: Enantioselective and Diastereoselective Conjugate Radical Additions to α-Arylidene Ketones and Lactones
    Supporting Information (PDF)
  • 2976
    Aldmairi, Abdul Hadi; Knight, David W.; Wirth, Thomas:

    Acid-Catalyzed Tandem Process for the One-Pot Synthesis of Oxazolidines

    Image for article: Acid-Catalyzed Tandem Process for the One-Pot Synthesis of Oxazolidines
    Supporting Information (PDF)

    • errata

  • e8
    Piras, Monica; Andriu, Alexandra; Testa, Andrea; Wienecke, Paul; Fleming, Ian N.; Zanda, Matteo:

    Design and Synthesis of an RGD Peptidomimetic-Paclitaxel Conjugate Targeting αvβ3 Integrin for Tumour-Directed Drug Delivery