DOI: 10.1055/s-00000131

Synfacts

Issue 08 · Volume 2010 · August 2010 DOI: 10.1055/s-002-21206

Synform

A64
Zanda, Matteo: SYNFORM ISSUE 2010/08

Synthesis of Natural Products and Potential Drugs

z851
All PDFs of this category
0851
Mañas, C. G.; Paddock, V. L.; Bochet, C. G.; Spivey, A. C.; White, A. J. P.; Mann, I.; Oppolzer, W.: Synthesis of (±)-Clivonine
0852
Endo, K.; Hirokami, M.; Shibata, T.: Synthesis of a Tamoxifen Homologue
0853
Han, K.; Kim, C.; Park, J.; Kim, M.-J.: Synthesis of (S)-Rivastigmine
0854
Sheikh, N. S.; Bataille, C. J.; Luker, T. J.; Brown, R. C. D.: Formal Synthesis of Eurylene
0855
Boone, M. A.; Tong, R.; McDonald, F. E.; Lense, S.; Cao, R.; Hardcastle, K. I.: Synthesis of ent-Abudinol B
0856
Yan et al., L.: Synthesis of MK-5596
0857
Weng, J.; Li, Y.-B.; Wang, R.-B.; Li, F.-Q.; Liu, C.; Chan, A. S. C.; Lu, G.: Synthesis of Oseltamivir
0858
Fischer, D. F.; Sarpong, R.: Synthesis of (+)-Complanadine A
0859
Huang, X.; O’Brien, E.; Thai, F.; Cooper, G.: Synthesis of RO5114436
0860
Hodgson, D. M.; Salik, S.; Fox, D. J.: Synthesis of (-)-Cubebol
0861
Friest, J. A.; Maezato, Y.; Broussy, S.; Blum, P.; Berkowitz, D. B.: Synthesis of (S)-Profens
0862
Martin, C. L.; Overman, L. E.; Rohde, J. M.: Synthesis of (-)-Actinophyllic Acid
0863
Yuan, C.; Chang, C.-T.; Axelrod, A.; Siegel, D.: Synthesis of (+)-Complanadine A
0864
Huang, X.; Broadbent, S.; Dvorak, C.; Zhao, S.-H.: Synthesis of the Core Structure of P2X7 Receptor Antagonists
0865
DelMonte, A. J.; Waltermire, R. E.; Fan, Y.; McLeod, D. D.; Gao, Z.; Gesenberg, K. D.; Girard, K. P.; Rosingana, M.; Wang, X.; Kuehne-Willmore, J.; Braem, A. D.; Castoro, J. A.: Synthesis of BMS-587101

Synthesis of Heterocycles

z867
All PDFs of this category
0867
Nakamura, I.; Zhang, D.; Terada, M.: Copper-Catalyzed Synthesis of Pyridine N-Oxides from α,β-Unsaturated Oximes
0868
Lu, J.; Gong, X.; Yang, H.; Fu, H.: Copper-Catalyzed One-Pot Synthesis of Benzimidazo[1,2-b]isoquinolin-11-ones
0869
Gaddam, V.; Ramesh, S.; Nagarajan, R.: CuI/La(OTf)3-Catalyzed Synthesis of Isomeric Ellipticine
0870
Moghaddam, F. M.; Mirjafary, Z.; Saeidian, H.; Taheri, S.; Soltanzadeh, B.: One-Step Synthesis of Annulated Hydroquinolines
0871
Chen, Z.; Zhu, J.; Xie, H.; Li, S.; Wu, Y.; Gong, Y.: Copper-Catalyzed Cascade Synthesis of Triazoloquinoxalines
0872
Varela-Fernández, A.; García-Yebra, C.; Varela, J. A.; Esteruelas, M. A.; Saá, C.: Osmium-Catalyzed Synthesis of 3-Benzoxepines
0873
Ye, Z.; Lv, G.; Wang, W.; Zhang, M.; Cheng, J.: Rhodium-Catalyzed Synthesis of 3-Aryl and 3-Alkenyl Phthalides
0874
Spiteri, C.; Mason, C.; Zhang, F.; Ritson, D. J.; Sharma, P.; Keeling, S.; Moses, J. E.: Synthesis of 1,2-Benzisoxazoles via a 1,3-Dipolar Cycloaddition
0875
Koldobskii, A. B.; Tsvetkov, N. P.; Solodova, E. V.; Kalinin, V. N.: A Lactonization Route to 5-(Trifluoromethyl)-2(5H)-furanones
0876
Liu, Y.; Bao, W.: Synthesis of 1,4-Benzodioxanes via Epoxide Opening and Cyclization
0877
Wahab, B.; Ellames, G.; Passey, S.; Watts, P.: Synthesis of Substituted Indoles Using Flow Microreactors
0878
Wang, H.-Y.; Mueller, D. S.; Sachwani, R. M.; Londino, H. N.; Anderson, L. L.: Synthesis of Pyrroles via [3,3]-Rearrangement and Paal-Knorr Reaction
0879
Volkova, Y. A.; Averina, E. B.; Grishin, Y. K.; Bruheim, P.; Kuznetsova, T. S.; Zefirov, N. S.: One-Step Synthesis 3-Nitroisoxazoles
0880
Wu, C.; Fang, Y.; Larock, R. C.; Shi, F.: Synthesis of 2H-Indazoles via [3+2]-Dipolar Cycloaddition
0881
Ueda, M.; Sato, A.; Ikeda, Y.; Miyoshi, T.; Naito, T.; Miyata, O.: Synthesis of Trisubstituted Isoxazoles via Gold-Catalyzed Domino Reaction

Synthesis of Materials and Unnatural Products

z883
All PDFs of this category
0883
Devaraj, N. K.; Hilderbrand, S.; Upadhyay, R.; Mazitschek, R.; Weissleder, R.: Turn-On Labeling in Living Cells
0884
Vadehra, G. S.; Wall, B. D.; Diegelmann, S. R.; Tovar, J. D.: Incorporation of π-Conjugated Molecules within Peptide Backbones
0885
Miyake, G. M.; Zhang, Y.; Chen, E. Y.-X.: Naturally Renewable Polymers from an Innovative Living Polymerization
0886
Caruso Jr., A.; Siegler, M. A.; Tovar, J. D.: Stable Borepin Rings
0887
Sun, Q.-F.; Iwasa, J.; Ogawa, D.; Ishido, Y.; Sato, S.; Ozeki, T.; Sei, Y.; Yamaguchi, K.; Fujita, M.: Emergent Self-Assembly
0888
Miki, K.; Fujita, M.; Inoue, Y.; Senda, Y.; Kowada, T.; Ohe, K.: Novel Cyclyne via Mild Reductive Aromatization
0889
Han, Y.-F.; Li, H.; Weng, L.-H.; Jin, G.-X.: C-H Activation Directed Multicomponent Assembly of Macrocycles
0890
Li, Y.; Li, C.; Yue, W.; Jiang, W.; Kopecek, R.; Qu, J.; Wang, Z.: Simple Perfluoroalkylation
0891
Collin, J.-P.; Durola, F.; Frey, J.; Heitz, V.; Reviriego, F.; Sauvage, J.-P.; Trolez, Y.; Rissanen, K.: A Cyclic [4]Rotaxane
0892
Chu, L.; Qing, F.-L.: Trifluoromethylation of Terminal Alkynes
0893
Lang, T.; Guenet, A.; Graf, E.; Kyritsakas, N.; Hosseini, M. W.: Porphyrin-Based Molecular Turnstiles
0894
Kung, Y.-H.; Cheng, Y.-S.; Tai, C.-C.; Liu, W.-S.; Shin, C.-C.; Ma, C.-C.; Tsai, Y.-C.; Wu, T.-C.; Kuo, M.-Y.; Wu, Y.-T.: Benzo[k]fluoranthenes
0895
Bonifácio, V. D. B.; Morgado, J.; Scherf, U.: Sticky Caps for Polymers
0896
Troshin, P. A.; Khakina, E. A.; Peregudov, A. S.; Konarev, D. V.; Soulimenkov, I. V.; Peregudova, S. M.; Lyubovskaya, R. N.: A Stable Fullerene Anion

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

z897
All PDFs of this category
0897
Chen, Q.-A.; Dong, X.; Chen, M.-W.; Wang, D.-S.; Zhou, Y.-G.; Li, Y.-X.: Diastereoselective Synthesis of Axially Chiral Bis-sulfoxide Ligands
0898
Wang, D.; Ye, X.; Shi, X.: Gold-Catalyzed Synthesis of E-α-Haloenones from Propargyl Acetates
0899
Malik, H. A.; Sormunen, G. J.; Montgomery, J.: Regiocontrol in the Nickel-Catalyzed Aldehyde-Alkyne Reductive Coupling
0900
Ito, J.-i.; Ujiie, S.; Nishiyama, H.: Chiral Bis(oxazolinyl)phenyl Ruthenium(II) Catalysts for Asymmetric Cyclopropanation
0901
Cho, H. Y.; Morken, J. P.: Nickel-Catalyzed Reductive Coupling of Dienes with Aldehydes
0902
Stenne, B.; Timperio, J.; Savoie, J.; Dudding, T.; Collins, S. K.: Construction of Chiral Tetrasubstituted Olefins Using Ring-Closing Metathesis
0903
Chen, M.; Roush, W. R.: E-Selective Allylboration of α-Substituted Allylboronates
0904
Luo, H.-K.; Woo, Y.-L.; Schumann, H.; Jacob, C.; van Meurs, M.; Yang, H.-Y.; Tan, Y.-T.: Synthesis and Application of C2-Bridged Diphosphine Palladium Complexes
0905
Fernández-Pérez, H.; Donald, S. M. A.; Munslow, I. J.; Benet-Buchholz, J.; Maseras, F.; Vidal-Ferran, A.: Modular Synthesis of P-OP Ligands and Application in Asymmetric Hydrogenation
0906
Ohmiya, H.; Yokokawa, N.; Sawamura, M.: Copper-Catalyzed Selective Aryl-Allyl Coupling
0907
He, L.; Liu, W.-J.; Ren, L.; Lei, T.; Gong, L.-Z.: Zirconium-Mediated Enantioselective Darzens Reaction
0908
Liu, H.; Du, D.-M.: Friedel-Crafts Alkylation of Indoles with Diphenylamine Bis(imidazoline) Ligands
0909
Xia, J.-B.; Liu, W.-B.; Wang, T.-M.; You, S.-L.: Ir-Catalyzed Asymmetric Allylic Amination and Pt-Catalyzed Cycloisomerization
0910
Yang, Z.; Wang, Z.; Bai, S.; Shen, K.; Chen, D.; Liu, X.; Lin, L.; Feng, X.: Scandium-Catalyzed Asymmetric α-Amination of 3-Substituted 2-Oxindoles
0911
Wang, C.; Han, Z.-Y.; Luo, H.-W.; Gong, L.-Z.: Selective Domino Synthesis of Heterocycles through Cooperative Catalysis
0912
Steurer, M.; Bolm, C.: Synthesis of Chiral Sulfonimidamides and Application in Asymmetric Henry Reaction
0913
Durán-Galván, M.; Connell, B. T.: Chromium-Catalyzed Enantioselective Synthesis of 1,3-Butadien-2-ylcarbinols
0914
Wu, J.; Chen, Y.; Panek, J. S.: Asymmetric Rh(II)- and Cu(I)-Catalyzed Si-H Insertion Leading to Chiral Crotylsilanes
0915
Herrmann, A. T.; Saito, T.; Stivala, C. E.; Tom, J.; Zakarian, A.: Synthesis of 1,3-syn-Diol Acetals via Re-Catalyzed Allylic Alcohol Transposition
0916
Tissot, M.; Müller, D.; Belot, S.; Alexakis, A.: Addition of Trialkylaluminium Regents to Extended Michael Acceptors
0917
Tiede, S.; Berger, A.; Schlesiger, D.; Rost, D.; Lühl, A.; Blechert, S.: Valine-Derived Ruthenium Complex for Catalytic Metathesis Desymmetrization
0918
Guo, F.; Lai, G.; Xiong, S.; Wang, S.; Wang, Z.: Friedel-Crafts Alkylation of Indoles via Combinatorial Transition-Metal Catalysis
0919
Fandrick, D. R.; Fandrick, K. R.; Reeves, J. T.; Tan, Z.; Tang, W.; Capacci, A. G.; Rodriguez, S.; Song, J. J.; Lee, H.; Yee, N. K.; Senanayake, C. H.: Enantioselective Propargylation of Aldehydes by Copper Catalysis
0920
Brak, K.; Ellman, J. A.: MIDA and BF3K in Rhodium-Catalyzed Stereoselective Addition to Aldimines
0921
Li, W. J.; Qiu, S. X.: A Novel Tetraoxazoline Ligand for Asymmetric Hydrosilylation
0922
Ito, H.; Toyoda, T.; Sawamura, M.: Sterospecific Copper-Catalyzed Formation of Cyclobutyl- and Cyclopentylboronates
0923
Luan, X.; Wu, L.; Drinkel, E.; Mariz, R.; Gatti, M.; Dorta, R.: Chemo- and Enantioselective Synthesis of 3-Allyl-3-aryl Oxindoles
0924
Reddy, B. V. S.; Borkar, P.; Chakravarthy, P. P.; Yadav, J. S.; Gree, R.: Synthesis of Heterobicycles by Intramolecular Aza-Prins Reaction
0925
Sun, X.; Li, W.; Zhou, L.; Zhang, X.: Enantioselective Hydrogenation of α-Dehydroamino Acid Esters
0926
Han, H.; Krische, M. J.: C-C Coupling of Ethanol and Dienes

Metal-Mediated Synthesis

z927
All PDFs of this category
0927
Sumida, Y.; Yorimitsu, H.; Oshima, K.: Nickel-Catalyzed Arylative Ring Opening
0928
Rao, M. L. N.; Banerjee, D.; Dhanorkar, R. J.: Atom-Efficient Coupling of Triarylbismuths with Bromide and Chloride Derivatives
0929
Clayden, J.; Donnard, M.; Lefranc, J.; Minassi, A.; Tetlow, D. J.: N-C Aryl Transfer via Umpolung Carbolithiation of Vinyl Ureas
0930
Kawano, T.; Hirano, K.; Satoh, T.; Miura, M.: Copper-Catalyzed Direct Amination of Azoles with Chloroamines at Room Temperature
0931
Tomioka, T.; Takahashi, Y.; Vaughan, T. G.; Yanase, T.: A One-Pot Synthesis of (Z)-Acrylonitriles via an α-Diaminoboryl Carbanion
0932
Kommidi, H.; Balasubramaniam, S.; Aidhen, I. S.: Synthetic Equivalents for the Preparation of 1,2,3,4-Tetrahydroisoquinolines
0933
Woerly, E. M.; Cherney, A. H.; Davis, E. K.; Burke, M. D.: Stereoretentive Suzuki-Miyaura Coupling of Haloallenes
0934
Sun, C.-L.; Wang, Y.; Zhou, X.; Wu, Z.-H.; Li, B.-J.; Guan, B.-T.; Shi, Z.-J.: Nickel-Catalyzed Synthesis of Poly-substituted Olefins from Alkenyl Acetates
0935
Bracegirdle, S.; Anderson, E. A.: Arylsilane Oxidation - New Routes to Hydroxylated Aromatics
0936
Rohbogner, C. J.; Wirth, S.; Knochel, P.: Phosphorodiamidate-Directed Metalation of N-Heterocycles using Mg- and Zn-TMP
0937
Abboud, M.; Mamane, V.; Aubert, E.; Lecomte, C.; Fort, Y.: Synthesis of 4,4′-Bipyridines via a Simple Dimerization Procedure
0938
Matsubara, R.; Jamison, T. F.: Nickel-Catalyzed Allylic Substitution of Simple Alkenes
0939
Tarr, J. C.; Johnson, J. S.: La(CN)3-Catalyzed Acyl Silane-Ketone Benzoin Addition
0940
Lundgren, R. J.; Peters, B. D.; Alsabeh, P. G.; Stradiotto, M.: A P,N-Ligand for the Palladium-Catalyzed Arylation of Ammonia
0941
Mikami, K.; Tomita, Y.; Itoh, Y.: Difluoromethylation of Lithium Enolates with Trifluoromethyl Iodide

Organo- and Biocatalysis

z943
All PDFs of this category
0943
Zhu, S.; Yu, S.; Wang, Y.; Ma, D.: Michael Addition of Aldehydes to 2-Amino-1-nitroethenes
0944
Yang, H.; Carter, R. G.: Enantioselective One-Pot Synthesis of Substituted Cyclohexenones
0945
Schmid, M. B.; Zeitler, K.; Gschwind, R. M.: NMR Detection of the Enamine Intermediate in Proline-Catalyzed Aldol Reactions
0946
Luo, S.; Zhou, P.; Li, J.; Cheng, J.-P.: Catalytic Asymmetric Retro-Aldol Reaction
0947
Čorić, I.; Vellalath, S.; List, B.: Catalytic Asymmetric Transacetalization
0948
Xiao, H.; Chai, Z.; Zheng, C.-W.; Yang, Y.-Q.; Liu, W.; Zhang, J.-K.; Zhao, G.: Asymmetric [3+2] Cycloaddition Catalyzed by 1,2-Aminophosphanes
0949
de Vincentiis, F.; Bencivenni, G.; Pesciaioli, F.; Mazzanti, A.; Bartoli, G.; Galzerano, P.; Melchiorre, P.: Aziridination of Cyclic Enones
0950
Blackmond, D. G.; Moran, A.; Hughes, M.; Armstrong, A.: Inversion of Enantioselectivity in Proline Catalysis by Basic Additives
0951
Phillips, E. M.; Roberts, J. M.; Scheidt, K. A.: NHC-Catalyzed Desymmetrization in Natural Product Synthesis
0952
Zhu, N.; Ma, B.-C.; Zhang, Y.; Wang, W.: Organocatalytic Vinylogous Mukaiyama Aldol Reactions
0953
Basak, A. K.; Shimada, N.; Bow, W. F.; Vicic, D. A.; Tius, M. A.: Bifunctional Catalysts for Asymmetric Nazarov Cyclizations
0954
Terrasson, V.; van der Lee, A.; de Figueiredo, R. M.; Campagne, J. M.: Cyclopropanation of α-Substituted α,β-Unsaturated Aldehydes
0955
Xue, F.; Lu, L.; Zhang, S.; Duan, W.; Wang, W.: Michael Reaction of α,α-Disubstituted Aldehydes and Maleimides
0956
Bernal, P.; Fernández, R.; Lassaletta, J. M.: Asymmetric Cyanosilylation of Nitroalkenes

Polymer-Supported Synthesis

z957
All PDFs of this category
0957
Arutyunyan, S.; Nefzi, A.: Solid-Phase Synthesis of Aminothiazoles
0958
Huang, Z.; Derksen, D. J.; Vederas, J. C.: Solid-Phase Synthesis of Peptides Using Cysteine Orthoesters
0959
Yan, G.; Jiang, Y.; Kuang, C.; Wang, S.; Liu, H.; Zhang, Y.; Wang, J.: Direct Borylation of Arenes Catalyzed by γ-Fe2O3
0960
Paira, R.; Paira, P.; Maity, A.; Mondal, S.; Hazra, A.; Sahu, K. B.; Naskar, S.; Saha, P.; Banerjee, M.; Mondal, N. B.: Synthesis of Fused Quinolinium Salts Using Amberlite IRA 402(OH)
0961
Ahmadibeni, Y.; Dash, C.; Grice, S. F. J. Le; Parang, K.: 5′-O-β,γ-Methylenetriphosphate Derivatives of Nucleosides
0962
Prastaro, A.; Ceci, P.; Chiancone, E.; Boffi, A.; Fabrizi, G.; Cacchi, S.: Protein-Stabilized Palladium Nanoparticles for Biaryl Coupling
0963
Colacino, E.; Villebrun, L.; Martinez, J.; Lamaty, F.: Ligand-Free Ullmann Arylation of Indole Using PEG3400-Cu2O-Cs2CO3
0964
Niknam, K.; Saberi, D.; Sefat, M. N.: Silica-Based S-Sulfonic Acid for the Strecker Synthesis
0965
Ding, F.; William, R.; Gorityala, B. K.; Ma, J.; Wang, S.; Liu, X.-W.: ZnCl2/Al2O3-Catalyzed Ferrier Azaglycosylation
0966
Lai, J.-J.; Salunke, D. B.; Sun, C.-M.: Microwave-Assisted Synthesis of Fused Quinoxalinones
0967
Singhal, S.; Jain, S. L.; Sain, B.: Oxidative Cyanation of Amines Using Heterogeneous Iron Phthalocyanines
0968
Kumar, A.; Akula, H. K.; Lakshman, M. K.: Simple Synthesis of Amides with Polymer-Supported Ph3P and Iodine
0969
Li, Y.; Giulionatti, M.; Houghten, R. A.: Silica-Phase Synthesis of Kahalalide B and Its Analogues

Addenda and Errata

0970
Expedient Total Synthesis of Kinamycin F
0970
Enantioselective Synthesis of Substituted Indanones