DOI: 10.1055/s-00000131

Synfacts

Issue 02 · Volume 2009 · February 2009 DOI: 10.1055/s-002-15179

Synform

A1

Synthesis of Natural Products and Potential Drugs

0117
0119
Burgey, C. S.; Paone, D. V.; Shaw, A. W.; Deng, J. Z.; Nguyen, D. N.; Potteiger, C. M.; Graham, S. L.; Vacca, J. P.; Williams, T. M.: Synthesis of Telcagepant (MK-0974)
0120
0121
Ebner, D. C.; Trend, R. M.; Genet, C.; McGrath, M. J.; O’Brien, P.; Stoltz, B. M.: Synthesis of (-)-Amurensinine
0122
Tiefenbacher, K.; Mulzer, J.: Formal Synthesis of (-)-Platencin
0123
Paterson, I.; Razzak, M.; Anderson, E. A.: Synthesis of Saliniketal B
0124
Navarro, I.; Basset, J.-F.; Hebbe, S.; Major, S. M.; Werner, T.; Howsham, C.; Bräckow, J.; Barrett, A. G. M.: Synthesis of 15G256β
0125
Takahashi, K.; Midori, M.; Kawano, K.; Ishihara, J.; Hatakeyama, S.: Synthesis of (-)-Salinosporamide A
0126
Varin, M.; Barré, E.; Iorga, B.; Guillou, C.: Synthesis of (±)-Codeine
0127
Sakakura, A.; Umemura, S.; Ishihara, K.: Synthesis of Fluvibactin
0128
Yun, S. Y.; Zheng, J.-C.; Lee, D.: Formal Synthesis of Platencin
0130
Cheung, L. L.; Marumoto, S.; Anderson, C. D.; Rychnovsky, S. D.: Synthesis of SCH 351448
0131
Guo, H.; Mortensen, M. S.; O’Doherty, G. A.: Formal Synthesis of RK-397

Synthesis of Heterocycles

0137
Fischer, D.; Tomeba, H.; Pahadi, N. K.; Patil, N. T.; Huo, Z.; Yamamoto, Y.: Synthesis of Isoquinolines by I2-Mediated Electrophilic Heteroannulation
0138
Feroci, M.; Chiarotto, I.; Rossi, L.; Inesi, A.: The Gewald Synthesis of 2-Aminothiophenes using Activated Sulfur
0139
Grigg, R.; Sridharan, V.; Shah, M.; Mutton, S.; Kilner, C.; MacPherson, D.; Milner, P.: Pd-Catalyzed Three-Component Synthesis of Isoindolones and Phthalazones
0140
Melkonyan, F.; Topolyan, A.; Yurovskaya, M.; Karchava, A.: Concise Cu-Catalyzed Synthesis of 3-Carboxyl-N-Aminoindoles
0141
Jordan-Hore, J. A.; Johansson, C. C. C.; Gulias, M.; Beck, E. M.; Gaunt, M. J.: Oxidative Pd(II)-Catalyzed C-H Bond Activation Route to Carbazoles
0145
0146
Ghosh, D.; Thander, L.; Ghosh, S. K.; Chattopadhyay, S. K.: Aza-Claisen-RCM Route to 1-Benzazepine Derivatives
0147

Synthesis of Materials and Unnatural Products

0149
Briquel, R.; Mazzolini, J.; Bris, T. Le; Boyron, O.; Boisson, F.; Delolme, F.; D’Agosto, F.; Boisson, C.; Spitz, R.: Functional End-Capping for PE
0150
Loudet, A.; Bandichhor, R.; Burgess, K.; Palma, A.; McDonnell, S. O.; Hall, M. J.; O’Shea, D. F.: Design and Synthesis of Near-IR Fluorophores
0151
Walker, W.; Veldman, B.; Chiechi, R.; Patil, S.; Bendikov, M.; Wudl, F.: Antiaromatic Lowering of the HOMO-LUMO Gap
0152
Shimizu, M.; Mochida, K.; Hiyama, T.: Silicon-Bridged Biaryls
0154
Feng, X.; Feng, F.; Yu, M.; He, F.; Xu, Q.; Tang, H.; Wang, S.; Li, Y.; Zhu, D.: Tyrosinase Activity Sensor
0155
Gug, S.; Bolze, F.; Specht, A.; Bourgogne, C.; Goeldner, M.; Nicoud, J.-F.: A Protecting Group for Two-Photon Uncaging
0156
Matsuo, Y.; Iwashita, A.; Abe, Y.; Li, C.-Z.; Matsuo, K.; Hashiguchi, M.; Nakamura, E.: Efficient Regioselective 1,4-Substitution of [60]Fullerenes
0157
Velasco, V. M.; Zolotukhin, M. G.; Guzmán-Gutiérrez, M. T.; Morales, S. L.; Fomine, S.; Carreón-Castro, M. P.; Salmón, M.; Scherf, U.: Aromatic Polymers with Pentafluorophenyl Groups
0159
Ralli, P.; Zhang, Y.; Lemal, D. M.: Perfluorobarrelene
0161
Riehm, T.; De Paoli, G.; Wadepohl, H.; De Cola, L.; Gade, L. H.: A Handle for Perylene Dyes

Metal-Catalyzed Asymmetric Synthesis and Stereoselective Reactions

0163
Kim, D. E.; Lee, B. H.; Rajagopalasarma, M.; Genêt, J.-P.; Ratovelomanana-Vidal, V.; Jeong, N.: Desymmetrization of Diallyl Acetals of Alkynals by Rodium Catalysis
0165
Shintani, R.; Park, S.; Shirozu, F.; Murakami, M.; Hayashi, T.: Palladium-Catalyzed Synthesis of Chiral Lactams from Racemic Lactones
0166
0168
Tan, C.; Liu, X.; Wang, L.; Wang, J.; Feng, X.: Asymmetric Aza-Henry Reaction of Ketoimines
0170
Qiu, M.; Hu, X.-P.; Huang, J.-D.; Wang, D.-Y.; Deng, J.; Yu, S.-B.; Duan, Z.-C.; Zheng, Z.: A New Phosphine-Aminophosphine Ligand for Enantioselective Hydrogenation
0171
Thu, H.-Y.; Tong, G. S.-M.; Huang, J.-S.; Chan, S. L.-F.; Deng, Q.-H.; Che, C.-M.: Selective Carbene Insertion into Primary C-H Bonds
0174
Li, Z.-W.; Wang, T.-L.; He, Y.-M.; Wang, Z.-J.; Fan, Q.-H.; Pan, J.; Xu, L.-J.: Synthesis of Chiral Tetrahydroquinolines by Asymmetric Hydrogenation
0176
Chen, I.-H.; Oisaki, K.; Kanai, M.; Shibasaki, M.: Copper(I)-Catalyzed Hetero-Diels-Alder Reaction of Ketones
0177
Du, Y.; Xu, L.-W.; Shimizu, Y.; Oisaki, K.; Kanai, M.; Shibasaki, M.: Copper-Catalyzed Asymmetric Reductive Mannich Reaction
0178
Morimoto, H.; Yoshino, T.; Yukawa, T.; Lu, G.; Matsunaga, S.; Shibasaki, M.: Lewis Base Assisted Brønsted Base: Phosphine Oxides and La-Aryloxides
0179
Hernández-Toribio, J.; Arrayás, R. G.; Carretero, J. C.: Copper-Catalyzed Mannich Reaction of Glycinate Schiff Bases with Imines
0180
0185
Bercot, E. A.; Caille, S.; Bostick, T. M.; Ranganathan, K.; Jensen, R.; Faul, M. M.: Quaternary Center Formation via Diastereoselective Arylation of Enolates
0187
Zhao, J.-F.; Tsui, H.-Y.; Wu, P.-J.; Lu, J.; Loh, T.-P.: In(III)-PyBox Complex Catalyzed Enantioselective Carbonyl-ene Reaction
0188
Li, Z.; Gao, Y.; Jiao, Z.; Wu, N.; Wang, D. Z.; Yang, Z.: A Protocol for Palladium(II)-Mediated Alkoxycarbonylation

Metal-Mediated Synthesis

0191
Wilson, D. A.; Wilson, C. J.; Rosen, B. M.; Percec, V.: Ni-Catalyzed One-Pot Neopentylglycol-borylation
0192
0194
0195
Berman, A. M.; Lewis, J. C.; Bergman, R. G.; Ellman, J. A.: Direct Arylation of α-Substituted Pyridines and Quinolines
0198
0201
Augustine, J. K.; Naik, Y. A.; Vairaperumal, V.; Narasimhan, S.: Di-tert-butyl Dicarbonate: A Versatile Carboxylating Agent
0203
Zhang, L.; Qing, J.; Yang, P.; Wu, J.: Hiyama Cross-Coupling of Aryl Mesylates

Organo- and Biocatalysis

0205
Uraguchi, D.; Asai, Y.; Ooi, T.: Organocatalytic Peptide Modification
0207
Hatano, M.; Maki, T.; Moriyama, K.; Arinobe, M.; Ishihara, K.: Chiral Brønsted Acid-Base Pyridinium Disulfonate Catalysts
0208
Lakhdar, S.; Tokuyasu, T.; Mayr, H.: Insights into Iminium Catalysis
0209
Graham, T. H.; Jones, C. M.; Jui, N. T.; MacMillan, D. W. C.: α-Alkylation of Aldehydes with Styrenes
0210
0211
Hayashi, Y.; Samanta, S.; Itoh, T.; Ishikawa, H.: Catalytic Asymmetric ”Aldol" Reaction
0213
Hahn, B. T.; Fröhlich, R.; Harms, K.; Glorius, F.: Proline Catalyzed anti-Selective Mannich Reaction
0216
0217
Chi, Y.; Scroggins, S. T.; Boz, E.; Fréchet, J. M. J.: Biomimetic Chemoselectivity Control of Aldol Reactions

Polymer-Supported Synthesis

0219
Ceylan, S.; Friese, C.; Lammel, C.; Mazac, K.; Kirschning, A.: Magnetic Nanoparticles as Inductive Heating Elements in Microreactors
0220
Motoyama, Y.; Abe, M.; Kamo, K.; Kosako, Y.; Nagashima, H.: Isomerization of Allyl Ethers with [Ru3]@SiEGcap
0221
Carrera, N.; Gutiérrez, E.; Benavente, R.; Villavieja, M. M.; Albéniz, A. C.; Espinet, P.: Clean Stille Reaction with Recyclable Stannylated Polynorbornenes
0222
Trilla, M.; Borja, G.; Pleixats, R.; Man, M. W. C.; Bied, C.; Moreau, J. J. E.: Silica-Supported Palladium Catalysts for Suzuki-Miyaura Reactions
0223
Kantam, M. L.; Chakravarti, R.; Chintareddy, V. R.; Sreedhar, B.; Bhargava, S.: Sequential Heck Coupling and Hydrogenation
0225
Monguchi, Y.; Kitamoto, K.; Ikawa, T.; Maegawa, T.; Sajiki, H.: C-N Coupling Reaction Catalyzed by Palladium on Carbon
0226
0228
0229
Pande, S.; Saha, A.; Jana, S.; Sarkar, S.; Basu, M.; Pradhan, M.; Sinha, A. K.; Saha, S.; Pal, A.; Pal, T.: Alcohol Oxidation with Resin-Immoblized Cu Nanocomposites
0230
Jiang, H.-y; Yang, C.-f; Li, C.; Fu, H.-y; Chen, H.; Li, R.-x; Li, X.-j: Asymmetric Hydrogenation of Ketones Using Ir/SiO2/Ph3P/Diamine Catalysts
0231
Sakai, H.; Tsutsumi, K.; Morimoto, T.; Kakiuchi, K.: Silica-Supported Palladium-Catalyzed Synthesis of Indole Derivatives